Histone Acetyltransferase Inhibitor II, p300/CBP HAT inhibitor (RMML-00120943)
Cat. No.: RMML-00120943
Category: Inhibitors & Activators
INQUIRY
10 mg
Selective, cell permeable p300/CBP HAT inhibitor
Product Features
| Source | Synthetic |
|---|---|
| Purity | > 98% |
| Key Features | Selective, cell permeable p300/CBP HAT inhibitor; CAS Number: 932749-62-7; Purity: > 98%; Soluble in DMSO to 100 mM and in ethanol to 25mM; Form / State: Solid; Source: Synthetic |
Compound Information
| Target Pathways | p300/CBP HAT |
|---|---|
| Biological Description | Selective, cell-permeable p300/CBP histone acetyltranserase inhibitor (IC50 = 5 μM). Antitumor agent. Active in vitro. |
| CAS Number | 932749-62-7 |
| Chemical Name | 2,6-Bis[(3-bromo-4-hydroxyphenyl)methylene]cyclohexanone |
| SMILES | Oc1ccc(cc1Br)/C=C3\CCC/C(=C\c2cc(Br)c(O)cc2)C3=O |
| Molecular Formula | C20H16Br2O3 |
| Molecular Weight | 464.15 Da |
| PubChem Identifier | 16203606 |
Storage & Shipping
| Handling | Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. |
|---|---|
| Solubility | Soluble in DMSO to 100 mM and in ethanol to 25 mM |
| Storage & Shipping | Store at 4°C. Store under desiccating conditions. The product can be stored for up to 12 months. |
For research use only. Not for clinical use.
