Ko-143, BCRP inhibitor (RMML-00120803)
Cat. No.: RMML-00120803
Category: Inhibitors & Activators
INQUIRY
5 mg
Potent, selective BCRP inhibitor
Product Features
| Source | Synthetic |
|---|---|
| Key Features | Potent, selective BCRP inhibitor; CAS Number: 461054-93-3; Soluble in ethanol to 100 mM and in DMSO to 50 mM; Form / State: Solid; Source: Synthetic |
Compound Information
| Target Pathways | BCRP |
|---|---|
| CAS Number | 461054-93-3 |
| Chemical Name | (3S,6S,12aS)-1,2,3,4,6,7,12,12a-Octahydro-9-methoxy-6-(2-methylpropyl)-1,4-dioxopyrazino[1',2':1,6]pyrido[3,4-b]indole-3-propanoic acid 1,1-dimethylethyl ester |
| SMILES | CC(C)C[C@H]1C2=C(C[C@@H]3N1C(=O)[C@@H](NC3=O)CCC(=O)OC(C)(C)C)C4=C(N2)C=C(C=C4)OC |
| Molecular Formula | C26H35N3O5 |
| Molecular Weight | 469.57 Da |
| PubChem Identifier | 10322450 |
Storage & Shipping
| Handling | Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. Refer to SDS for further information. |
|---|---|
| Solubility | Soluble in ethanol to 100 mM and in DMSO to 50 mM |
| Storage & Shipping | Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months. |
For research use only. Not for clinical use.
