PF-3758309 (RMML-00120064)
Cat. No.: RMML-00120064
Category: Inhibitors & Activators
INQUIRY
5 mg
A potent small molecule inhibitor of PAK4
Product Features
| Purity | ≥ 98% |
|---|---|
| Key Features | A potent small molecule inhibitor of PAK4; CAS Number: 898044-15-0; Purity: ≥ 98%; Soluble to in DMSO to 10 mM; Form / State: Solid |
Compound Information
| Biological Description | A potent small molecule inhibitor of p21-activated kinase 4 (PAK4) with potential antineoplastic activity. It binds to PAK4, inhibiting PAK4 activity and cancer cell growth. PAK4, a serine/threonine kinase belonging to the p21-activated kinase (PAK) family, is often upregulated in a variety of cancer cell types and plays an important role in cancer cell motility, proliferation, and survival. |
|---|---|
| Alternative Names | 898044-15-0, UNII-PK459EA5I2 |
| CAS Number | 898044-15-0 |
| Chemical Name | N-[(1S)-2-(dimethylamino)-1-phenylethyl]-6,6-dimethyl-3-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]-1,4-dihydropyrrolo[3,4-c]pyrazole-5-carboxamide |
| SMILES | CC1=NC2=C(C(=N1)NC3=NNC4=C3CN(C4(C)C)C(=O)NC(CN(C)C)C5=CC=CC=C5)SC=C2 |
| Molecular Formula | C25H30N8OS |
| Molecular Weight | 490.60 Da |
| PubChem Identifier | 25227462 |
Storage & Shipping
| Handling | Toxic, refer to SDS for further information. |
|---|---|
| Solubility | Soluble to in DMSO to 10 mM |
| Storage & Shipping | Shipped at 4°C. Store at -20°C long term. Store in the dark. |
For research use only. Not for clinical use.
