SR 27897 (Lintitript), CCK1 receptor antagonist (RMML-00120399)
Cat. No.: RMML-00120399
Category: Inhibitors & Activators
INQUIRY
50 mg
10 mg
Highly potent, selective, competitive, non-peptide CCK1 receptor antagonist
Product Features
| Source | Synthetic |
|---|---|
| Purity | > 98% |
| Key Features | Highly potent, selective, competitive, non-peptide CCK; 1; receptor antagonist; CAS Number: 136381-85-6; Purity: > 98%; Soluble in DMSO to 100 mM; Form / State: Solid; Source: Synthetic |
Compound Information
| Target Pathways | CCK1 receptor |
|---|---|
| Biological Description | Highly potent, selective, competitive, non-peptide CCK1 receptor antagonist (Ki = 0.2 nM). Increases plasma leptin levels. Shows central effects. Stimulates food intake in vivo. Orally active. |
| CAS Number | 136381-85-6 |
| Chemical Name | 2-[[[4-(2-Chlorophenyl)-2-thiazolyl]amino]carbonyl]-1H-indole-1-acetic acid |
| SMILES | O=C(Nc1nc(cs1)c2ccccc2Cl)c4cc3ccccc3n4CC(=O)O |
| Molecular Formula | C20H14ClN3O3S |
| Molecular Weight | 411.86 Da |
| PubChem Identifier | 122077 |
Storage & Shipping
| Handling | Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour. |
|---|---|
| Solubility | Soluble in DMSO to 100 mM |
| Storage & Shipping | Store at 4°C. The product can be stored for up to 12 months. |
For research use only. Not for clinical use.
